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Descriptor English: Ketanserin
Descriptor Spanish: Ketanserina
Descriptor ketanserina
Scope note: Antagonista selectivo de receptores de serotonina que posee propiedades débiles como bloqueante de receptores adrenérgicos. Esta sustancia es efectiva para reducir la presión sanguínea en los casos de hipertensión esencial. Asimismo, es antiagregante plaquetario. Tiene buena tolerancia y es particularmente efectiva en los pacientes de edad.
Descriptor Portuguese: Ketanserina
Descriptor French: Kétansérine
Entry term(s): R 41 468
R-41 468
R-41,468
R41 468
R41,468
R41468
Tree number(s): D03.383.621.365
D03.633.100.786.830.333
RDF Unique Identifier: https://id.nlm.nih.gov/mesh/D007650
Scope note: A selective serotonin receptor antagonist with weak adrenergic receptor blocking properties. The drug is effective in lowering blood pressure in essential hypertension. It also inhibits platelet aggregation. It is well tolerated and is particularly effective in older patients.
Allowable Qualifiers: AA analogues et dérivés
AD administration et posologie
AE effets indésirables
AG agonistes
AI antagonistes et inhibiteurs
AN analyse
BL sang
CF liquide cérébrospinal
CH composition chimique
CL classification
CS synthèse chimique
EC économie
HI histoire
IM immunologie
IP isolement et purification
ME métabolisme
PD pharmacologie
PK pharmacocinétique
PO intoxication
RE effets des radiations
SD ressources et distribution
ST normes
TO toxicité
TU usage thérapeutique
UR urine
Pharm Action: Antihypertensive Agents
Platelet Aggregation Inhibitors
Serotonin Antagonists
Registry Number: 97F9DE4CT4
CAS Type 1 Name: 2,4(1H,3H)-Quinazolinedione, 3-(2-(4-(4-fluorobenzoyl)-1-piperidinyl)ethyl)-
DeCS ID: 19223
Unique ID: D007650
Documents indexed in the Virtual Health Library (VHL): Click here to access the VHL documents
Date Established: 1987/01/01
Date of Entry: 1986/04/09
Revision Date: 2016/05/31
Kétansérine - Preferred
Concept UI M0011983
Preferred term Kétansérine
R-41,468 - Narrower
Concept UI M0353421
Preferred term R-41,468
Entry term(s) R 41 468
R-41 468
R41 468
R41,468
R41468



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